CGP 20712A, CAS 105737-62-0

Formulation: A solid

Formal Name: 2-hydroxy-5-[2-[[2-hydroxy-3-[4-[1-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl]phenoxy]propyl]amino]ethoxy]-benzamide, monomethanesulfonate

Purity: ≥95%

Formula Markup: C23H25F3N4O5 • CH3SO3H

Formula Weight: 590,6

Shelf life (days): 1460

CAS Number: 105737-62-0

Notes: CGP 20712A is an antagonist of the β1-adrenergic receptor (β1-AR; IC50 = 0.7 nM).{49844} It is selective for β1-ARs over β2-ARs (IC50 = 6,700 nM). CGP 20712 A (0.1-1,000 µM) inhibits adenylyl cyclase activity induced by the β1- and β2-AR agonist isoproterenol (Item No. 15592) in brown adipose tissue plasma membranes isolated from both lean and pre-obese rat pups.{49845}

• SKU: CAY40765-1
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 40765-1
• Package Unit: 1 mg
• Quantity Unit: STK