CID-5157334, CAS 651295-98-6

Formulation: A solid

Formal Name: 2,4-dichloro-N-[4-[(phenylamino)sulfonyl]phenyl]-benzamide

Purity: ≥95%

Formula Markup: C19H14Cl2N2O3S

Formula Weight: 421,3

Shelf life (days): 1460

CAS Number: 651295-98-6

Notes: CID-5157334 is a surrogate agonist of G protein-coupled receptor 27 (GPR27).{54081} It induces recruitment of β-arrestin-2 in complementation assays using wild-type GPR27 or a GPR27-vasopressin 2 (GPR27V2) chimeric receptor (EC50s = 7.943 and 0.417 nM, respectively) but does not induce recruitment of β-arrestin-1 in the same assay or activation of the Gq, Gs, or Gi signaling pathways in aequorin-GFP assays. CID-5157334 is selective for GPR27 over GPR85V2 and GPR173V2 chimeric receptors at 15 µM.

• SKU: CAY41677-25
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 41677-25
• Package Unit: 25 mg
• Quantity Unit: STK