Dexloxiglumide, CAS 119817-90-2

Formulation: A solid

Formal Name: (4R)-4-[(3,4-dichlorobenzoyl)amino]-5-[(3-methoxypropyl)pentylamino]-5-oxo-pentanoic acid

Purity: ≥98%

Formula Markup: C21H30Cl2N2O5

Formula Weight: 461,4

Shelf life (days): 1460

CAS Number: 119817-90-2

Notes: Dexloxiglumide is a cholecystokinin (CCK) receptor antagonist and is the single (R) isomer of loxiglumide (Item No. 25534).{61608,61609} It selectively binds to the CCK1 receptor over CCK2 in CHO cells expressing the rat receptors (Kis = 0.0234 and 5.88 µM, respectively).{61608} Dexloxiglumide (20 µmol/kg) inhibits guinea pig gallbladder contractions induced by the CCK agonist CCK octapeptide (sulfated) (CCK-8S; Item No. 23371). It reduces CCK-8-induced gastric emptying in rats (ID50 = 1.14 mg/kg).{61609}

• SKU: CAY34759-25
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 34759-25
• Green Labware: No
• Package Unit: 25 mg
• Quantity Unit: STK