GSK1702934A, CAS 924377-85-5

Formulation: A solid

Formal Name: 1,3-dihydro-1-[1-[(5,6,7,8-tetrahydro-4H-cyclohepta[b]thien-2-yl)carbonyl]-4-piperidinyl]-2H-benzimidazol-2-one

Purity: ≥98%

Formula Markup: C22H25N3O2S

Formula Weight: 395,5

Shelf life (days): 1460

CAS Number: 924377-85-5

Notes: GSK1702934A is an activator of transient receptor potential canonical 3 (TRPC3) and TRPC6.{58569} It induces TRPC3- and TRPC6-dependent currents in whole-cell patch-clamp assays using HEK293 cells expressing the human channels (EC50s = 0.08 and 0.44 µM, respectively). GSK1702934A enhances contractility and induces arrhythmias in hearts isolated from TRPC3-overexpressing, but not wild-type, mice.{58570}

• SKU: CAY34576-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 34576-5
• Green Labware: No
• Package Unit: 5 mg
• Quantity Unit: STK