Imidafenacin, CAS 170105-16-5

Formulation: A solid

Formal Name: 2-methyl-α,α-diphenyl-1H-imidazole-1-butanamide

Purity: ≥98%

Formula Markup: C20H21N3O

Formula Weight: 319,4

Shelf life (days): 1460

CAS Number: 170105-16-5

Notes: Imidafenacin is an antagonist of muscarinic acetylcholine receptors (mAChRs; Kis = 7.55, 22.6, 1.42, 8.86, and 2.63 nM, respectively, for recombinant human M1-M5 receptors).{66499} It binds to isolated guinea pig bladders (Kb = 0.813 nM) and inhibits ACh release from isolated rat bladders (IC50 = 0.747 nM). Imidafenacin (10-300 µg/kg) reduces urine volume in orally water-loaded rats.{66500} Formulations containing imidafenacin have been used in the treatment of overactive bladder.

• SKU: CAY37420-25
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 37420-25
• Green Labware: No
• Package Unit: 25 mg
• Quantity Unit: STK