Immethridine (hydrobromide), CAS 699020-93-4

Formulation: A solid

Formal Name: 4-(1H-imidazol-5-ylmethyl)-pyridine, dihydrobromide

Purity: ≥98%

Formula Markup: C9H9N3 • 2HBr

Formula Weight: 321

Shelf life (days): 1460

CAS Number: 699020-93-4

Notes: Immethridine is a potent histamine H3 receptor agonist (Ki = 0.85 nM).{46585} It is selective for histamine H3 over histamine H4 receptors (Ki = 245 nM). Immethridine inhibits cAMP-stimulated β-galactosidase transcription in SK-N-MC cells expressing human H3 receptors (EC50 = 0.18 nM) and induces a concentration-dependent decrease of the electrically induced twitch contraction in isolated guinea pig ileum. In vivo, immethridine (30 mg/kg, s.c.) inhibits hydrochloric acid-induced formation of gastric lesions in rats.{46586}

• SKU: CAY29502-1
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 29502-1
• Green Labware: No
• Package Unit: 1 mg
• Quantity Unit: STK