JTC 801, CAS 244218-51-7

Formulation: A crystalline solid

Formal Name: N-(4-amino-2-methyl-6-quinolinyl)-2-[(4-ethylphenoxy)methyl]-benzamide, monohydrochloride

Purity: ≥98%

Formula Markup: C26H25N3O2 • HCl

Formula Weight: 448

Shelf life (days): 1460

CAS Number: 244218-51-7

Notes: JTC 801 is an antagonist of the nociceptin receptor (ORL1; Ki = 44.5 nM; IC50 = 94 nM) that is >100-, >100-, and >3-fold more selective for ORL1 over the related δ-, κ-, and µ-opioid receptors, respectively.{33471} It demonstrates anti-nociceptive effects in acute pain models in mice upon oral administration at 1 mg/kg.{33471}

• SKU: CAY21254-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 21254-10
• Green Labware: No
• Package Unit: 10 mg
• Quantity Unit: STK