L-368,899 (hydrochloride), CAS 160312-62-9

Formulation: A solid

Formal Name: [1S-[1α,2α(R*),4β]]-2-amino-N-[7,7-dimethyl-1-[[[4-(2-methylphenyl)-1-piperazinyl]sulfonyl]methyl]bicyclo[2.2.1]hept-2-yl]-4-(methylsulfonyl)-butanamide, monohydrochloride

Purity: ≥98%

Formula Markup: C26H42N4O5S2 • HCl

Formula Weight: 591,2

Shelf life (days): 1460

CAS Number: 160312-62-9

Notes: L-368,899 is a non-peptide oxytocin receptor antagonist (IC50s = 8.9 and 26 nM in radioligand binding assays using isolated human and rat uterus, respectively).{53545} It is selective for oxytocin receptors over vasopressin V1a and V2 receptors (IC50s = 370 and 570 nM, respectively). L-368,899 reduces oxytocin-induced contraction of isolated rat uterus (pA2 = 8.9) and in situ rat uterus (ED50 = 0.35 mg/kg, i.v.).

• SKU: CAY29868-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 29868-5
• Green Labware: No
• Package Unit: 5 mg
• Quantity Unit: STK