MIPS521, CAS 1146188-19-3

Formulation: A solid

Formal Name: [2-amino-4-[3,5-bis(trifluoromethyl)phenyl]-3-thienyl](4-chlorophenyl)-methanone

Purity: ≥98%

Formula Markup: C19H10ClF6NOS

Formula Weight: 449,8

Shelf life (days): 1460

CAS Number: 1146188-19-3

Notes: MIPS521 is an adenosine A1 receptor positive allosteric modulator.{49809} It binds to adenosine A1 receptors (Kb = 11 µM) and enhances adenosine-induced inhibition of forskolin-induced cAMP production in CHO cells expressing recombinant human adenosine A1 receptors when used at concentrations ranging from 0.3 to 30 µM. In vivo, MIPS521 (10 and 30 µg/animal) increases the mechanical paw withdrawal threshold in a rat model of neuropathic pain induced by partial sciatic nerve ligation.

• SKU: CAY37776-10
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 37776-10
• Package Unit: 10 mg
• Quantity Unit: STK