PSB-KD107, CAS 955121-65-0

Formulation: A crystalline solid

Formal Name: 6,7,8,9-tetrahydro-9-[2-(1H-indol-3-yl)ethyl]-1,3-dimethyl-pyrimido[2,1-f]purine-2,4(1H,3H)-dione

Purity: ≥98%

Formula Markup: C20H22N6O2

Formula Weight: 378,4

Shelf life (days): 730

CAS Number: 955121-65-0

Notes: PSB-KD107 is an agonist of the orphan G protein-coupled receptor GPR18 (EC50 = 0.56 µM in a β-arrestin recruitment assay using CHO cells expressing the human receptor).{58090,44024} It is selective for GPR18 over GPR55, as well as cannabinoid 1 (CB1) and CB2 receptors, at 10 µM but also binds to the adenosine A2A receptor (Ki = 0.33 µM for the rat receptor).{58090,58091}

• SKU: CAY31393-1
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 31393-1
• Green Labware: No
• Package Unit: 1 mg
• Quantity Unit: STK