RO5028442, CAS 920022-47-5

Formulation: A crystalline solid

Formal Name: [6-chloro-1-[2-(dimethylamino)ethyl]-1H-indol-3-yl]spiro[isobenzofuran-1(3H),4′-piperidin]-1′-yl-methanone

Purity: ≥98%

Formula Markup: C25H28ClN3O2

Formula Weight: 438

Shelf life (days): 1460

CAS Number: 920022-47-5

Notes: RO5028442 is a brain-penetrant antagonist of vasopressin V1a receptors (Kis = 1 and 39 nM for the human and mouse receptors, respectively).{58074} It is greater than 30,000-fold selective for V1 over V2 receptors, as well as over a panel of 120 receptors, ion channels, and enzymes at 3 µM.

• SKU: CAY31452-100
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 31452-100
• Green Labware: No
• Package Unit: 100 mg
• Quantity Unit: STK