SKF 82958 (hydrobromide), CAS 74115-01-8

Formulation: A solid

Formal Name: 6-chloro-2,3,4,5-tetrahydro-1-phenyl-3-(2-propen-1-yl)-1H-3-benzazepine-7,8-diol, monohydrobromide

Purity: ≥98%

Formula Markup: C19H20ClNO2 • HBr

Formula Weight: 410,7

Shelf life (days): 1460

CAS Number: 74115-01-8

Notes: SKF 82958 is a dopamine D1 receptor agonist (K0.5 = 4 nM in a radioligand binding assay).{45668} It is selective for dopamine D1 over D2 receptors (K0.5 = 73 nM). SKF 82958 induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50 = 491 nM). SKF 82958 (3 mg/kg) prevents and reverses fentanyl-induced respiratory depression, without affecting analgesia, in cats.{45669} It also increases locomotion and rearing in rats.{45670}

• SKU: CAY29033-25
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 29033-25
• Green Labware: No
• Package Unit: 25 mg
• Quantity Unit: STK