TFLLR-NH2 (trifluoroacetate salt)

Formulation: A solid

Formal Name: (S)-2-((S)-2-((2S,3R)-2-amino-3-hydroxybutanamido)-3-phenylpropanamido)-N-((S)-1-(((S)-1-amino-5-guanidino-1-oxopentan-2-yl)amino)-4-methyl-1-oxopentan-2-yl)-4-methylpentanamide, trifluoroacetate salt

Purity: ≥98%

Formula Markup: C31H53N9O6 • XCF3COOH

Formula Weight: 647,8

Shelf life (days): 1460

Notes: TFLLR-NH2 is a synthetic peptide agonist of proteinase-activated receptor 1 (PAR1) that induces calcium mobilization in isolated rat dorsal root ganglion neurons (EC50 = 1.9 μM).{51082} In vivo, TFLLR-NH2 (3 μmol/kg) stimulates plasma extravasation in the bladder, esophagus, stomach, intestine, and pancreas in wild-type, but not PAR1-/-, mice. It also reduces carrageenan-induced hyperalgesia in rats.{51083}

• SKU: CAY27548-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 27548-5
• Green Labware: No
• Package Unit: 5 mg
• Quantity Unit: STK