UCSF924, CAS 1434515-70-4

Formulation: A solid

Formal Name: 6-methyl-2-[[(3-phenoxypropyl)amino]methyl]-4-quinolinol

Purity: ≥98%

Formula Markup: C20H22N2O2

Formula Weight: 322,4

Shelf life (days): 1460

CAS Number: 1434515-70-4

Notes: UCSF924 is a dopamine D4 receptor agonist.{67821} It selectively induces β-arrestin translocation over Gαi/o signaling in HEK293T cells expressing human dopamine D4 receptors by 7.4-fold at 1 µM. UCSF924 selectively induces cAMP accumulation in HEK293T cells expressing human dopamine D4 receptors (EC50 = 4.2 nM) over HEK293T cells expressing human dopamine D2 or dopamine D3 receptors (EC50s = >10 µM for both) and induces β-arrestin recruitment in HTLA cells expressing human dopamine D4 receptors over a panel of HTLA cells expressing one of 320 non-olfactory G protein-coupled receptors (GPCRs) at 1 µM.

• SKU: CAY41317-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 41317-5
• Package Unit: 5 mg
• Quantity Unit: STK