VCP171, CAS 1018830-99-3

Formulation: A crystalline solid

Formal Name: [2-amino-4-[3-(trifluoromethyl)phenyl]-3-thienyl]phenyl-methanone

Purity: ≥98%

Formula Markup: C18H12F3NOS

Formula Weight: 347,4

Shelf life (days): 730

CAS Number: 1018830-99-3

Notes: VCP171 is a positive allosteric modulator of adenosine A1 receptors (EC50 = 15.8 μM in a kinetic assay measuring agonist dissociation).{61017}. It reduces AMPA receptor-mediated evoked excitatory postsynaptic currents (eEPSCs) in lamina I and lamina II neurons in a rat model of neuropathic pain (EC50s = 1.995 and 0.251 μM, respectively) to a greater extent than in sham control animals (EC50s = 2.512 and 0.631 μM, respectively).{45812}

• SKU: CAY30309-25
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 30309-25
• Green Labware: No
• Package Unit: 25 mg
• Quantity Unit: STK