MRS1220, CAS 183721-15-5

Formulation: A solid

Formal Name: N-[9-chloro-2-(2-furanyl)[1,2,4]triazolo[1,5-c]quinazolin-5-yl]-benzeneacetamide

Purity: ≥95%

Formula Markup: C21H14ClN5O2

Formula Weight: 403,8

Shelf life (days): 1460

CAS Number: 183721-15-5

Notes: MRS1220 is an adenosine A3 receptor antagonist (Ki = 0.65 nM for the human receptor).{69827} It is selective for human adenosine A3 receptors over rat adenosine A1 and A2receptors (Kis = 305 and 52 nM, respectively). MRS1220 inhibits [35S]GTPγS binding in HEK293 cells expressing human adenosine A3 receptors (IC50 = 7.2 nM). In vivo, MRS1220 (0.15 mg/kg) decreases tumor growth and angiogenesis in a rat C6 glioma model.{69828}

• SKU: CAY41015-5
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 41015-5
• Package Unit: 5 mg
• Quantity Unit: STK