CGS 8216, CAS 77779-60-3

Product Description: CGS 8216 is a non-benzodiazepine brain benzodiazepine receptor ligand that binds to rat forebrain membranes with high affinity and specificity. CGS 8216 also inhibits 3H-flunitrazepam (3H-FLU) binding to rat synaptosomal membranes and blocks 3H-FLU labeling of brain benzodiazepine receptors in vivo with potency equivalent to Diazepam[1].

Applications: Neuroscience-Neuromodulation

Formula: C16H11N3O

References: [1]Czernik A J, Petrack B, Kalinsky H J, et al. CGS 8216: Receptor binding characteristics of a potent benzodiazepine antagonist[J]. Life sciences, 1982, 30(4): 363-372.

CAS Number: 77779-60-3

Molecular Weight: 261.28

Research Area: Neurological Disease

Target: GABA Receptor

• SKU: MEXHY-121116-5
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-121116-5
• Package Unit: 5 mg
• Quantity Unit: STK