BRD7-IN-2

Product Description: BRD7-IN-2 (compound 2-77) is a potent inhibitor of bromodomain-containing protein 7 (BRD7), targeting to prostate cancer cells. BRD7-IN-2 is selective for BRD7 rather than BRD9, with IC50s of 5.4 μM, and >300 μM, respectively.

Formula: C18H18N2O3

References: [1]Ordonez-Rubiano SC, Maschinot CA, Wang S, Sood S, Baracaldo-Lancheros LF, Strohmier BP, McQuade AJ, Smith BC, Dykhuizen EC. Rational Design and Development of Selective BRD7 Bromodomain Inhibitors and Their Activity in Prostate Cancer. J Med Chem. 2023 Aug 24;66(16):11250-11270.

Molecular Weight: 310.35

Compound Purity: 99.21

Research Area: others

Solubility: DMSO : 10 mg/mL (ultrasonic)

Target: Epigenetic Reader Domain

• SKU: MEXHY-149420-5
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-149420-5
• Green Labware: No
• Package Unit: 5 mg
• Quantity Unit: STK