Product Description: C3TD879 is a potent Type I kinase inhibitor. C3TD879 inhibits CITK catalytic activity with an IC50 of 12 nM[1].
Formula: C22H28N4O
References: [1]Maw JJ, et al. Discovery and Characterization of Selective, First-in-Class Inhibitors of Citron Kinase. J Med Chem. 2024 Feb 22;67(4):2631-2666.