CL 316243, CAS 138908-40-4

Description: CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate. CL316243 has the potential for the treatment obesity, diabetes and urge urinary incontinence.

CAS Number: 138908-40-4

Formula: C20H18ClNNa2O7

Molecular Weight: 465,79

References: Bloom JD, et al. Disodium (R,R)-5-[2-[[2-(3-chlorophenyl)-2-hydroxyethyl]-amino] propyl]-1,3-benzodioxole-2,2-dicarboxylate (CL 316,243). A potent beta-adrenergic agonist virtually specific for beta 3 receptors. A promising antidiabetic and antiobesity agent.J Med Chem. 1992 Aug 7;35(16):3081-4.

• SKU: TGMT10830-1mg
• Manufacturer: TargetMol Chemicals
• Manufacturer SKU: T10830-1mg
• Package Unit: 1 mg
• Quantity Unit: STK