EZH2-IN-18, CAS 2826234-37-9

Product Description: EZH2-IN-18 (compound 9e) is a potent inhibitor of enhancer of zeste homologue 2 (EZH2WT) with the IC50 of 1.01 nM. EZH2-IN-18 shows inhibition in proliferation and induction in apoptosis in tumor cells[1].

Formula: C24H20BrN3O3

References: [1]Jin Cai, et al. Design, synthesis and activity evaluation of quinolinone derivatives as EZH2 inhibitors. Bioorg Med Chem Lett. 2024 Jun 1:105:129726.

CAS Number: 2826234-37-9

Molecular Weight: 478.34

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Histone Methyltransferase

• SKU: MEXHY-161419-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-161419-0
• Green Labware: No
• Package Unit: Get quote
• Quantity Unit: STK