Galectin-3-IN-4, CAS 2496515-38-7

Product Description: Galectin-3-IN-4 (compound 5) is a carboxamide analog. Galectin-3-IN-4 is a potent, selective, and orally bioavailable inhibitor of human and mouse galectin-3, with IC50 values of 21 and 167 nM for hGal-3 and mGal-3, respectively. Galectin-3-IN-4 has IC50 values of 1580 and 2750 nM for hGal-1 and hGal-9, respectively[1].

Applications: Cancer-programmed cell death

Formula: C24H22ClF2N5O5S

References: [1]Liu C, et al. Identification of benzothiazole derived monosaccharides as potent, selective, and orally bioavailable inhibitors of human and mouse galectin-3; a rare example of using a S···O binding interaction for drug design. Bioorg Med Chem. 2024 Mar 1;101:117638.

CAS Number: 2496515-38-7

Molecular Weight: 565.98

Research Area: Cancer

Solubility: 10 mM in DMSO

Target: Galectin

• SKU: MEXHY-163407-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-163407-0
• Green Labware: No
• Package Unit: Get quote
• Quantity Unit: STK