Product Description: KDU731, an orally active C. parvum PI4K inhibitor with an IC50 value of 25 nM, blocks Cryptosporidium infection in vitro and in vivo[1][2]. KDU731 is a promising agent candidate for the treatment of diarrhea caused by Cryptosporidium and meets a broad range of safety[2].
Applications: Neuroscience-Neuromodulation
Formula: C22H16N6O2
References: [1]Ward HD, et al. New Tools for Cryptosporidium Lead to New Hope for Cryptosporidiosis. Trends Parasitol. 2017 Sep;33(9):662-664./[2]Manjunatha UH, et al. A Cryptosporidium PI(4)K inhibitor is a drug candidate for cryptosporidiosis. Nature. 2017 Jun 15;546(7658):376-380.
CAS Number: 1610610-48-4
Molecular Weight: 396.40
Compound Purity: 98.0
Research Area: Infection
Solubility: DMSO : 83.33 mg/mL (ultrasonic)
Target: Parasite;PI4K