Product Description: Myosin modulator 1 (Compound B141) is a modulator for myosin, that inhibits ATPase in rabbits psoas, porcine atria and in porcine ventricle, with IC25s of 0.42, 0.13 and 3.09 μM, respectively. Myosin modulator 1 regulates systolic cardiac performance in Sprague Dawley rats[1].
Formula: C18H14F3N5O2
References: [1]Hawryluk N, et al., 1,4-dihydroquinazolinone compounds and uses thereof. WO2024073426A1.
CAS Number: 3034189-56-2
Molecular Weight: 389.33
Research Area: Cardiovascular Disease
Solubility: 10 mM in DMSO
Target: Myosin