Tazemetostat, CAS 1403254-99-8

Description: Tazemetostat (EPZ6438) is a histone methyltransferase EZH2 inhibitor (IC50=11 nM) that is orally active, selective, and SAM-competitive. Tazemetostat exhibits antitumor activity and may be used for the treatment of epithelioid sarcoma/follicular lymphoma.

CAS Number: 1403254-99-8

Formula: C34H44N4O4

Molecular Weight: 572,74

References: Kawano S, et al. Preclinical Evidence of Anti-Tumor Activity Induced by EZH2 Inhibition in Human Models of Synovial Sarcoma. PLoS One. 2016 Jul 8;11(7):e0158888.

• SKU: TGMT1788-200mg
• Manufacturer: TargetMol Chemicals
• Manufacturer SKU: T1788-200mg
• Package Unit: 200 mg
• Quantity Unit: STK