TbPTR1 inhibitor 2, CAS 17557-67-4

Product Description: TbPTR1 inhibitor 2 (Compound 3a) is a PTR1 enzyme inhibitor, with IC50s of 34.2 and 32.9 μM for TbPTR1 and LmPTR1. TbPTR1 inhibitor 2 has anti-parasitic activity against T. brucei (IC50: 34.2 μM)[1].

Applications: COVID-19-immunoregulation

Formula: C8H8N2O2S2

References: [1]Linciano P, et al. Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections. J Med Chem. 2019 Apr 25;62(8):3989-4012.

CAS Number: 17557-67-4

Molecular Weight: 228.29

Compound Purity: 99.63

Research Area: Infection

Solubility: DMSO : 125 mg/mL (ultrasonic)

Target: Parasite

• SKU: MEXHY-W009689-100
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-W009689-100
• Green Labware: No
• Package Unit: 100 mg
• Quantity Unit: STK