α2A-AR agonist 1, CAS 2971825-58-6

Product Description: α2A-AR agonist 1 (Compound B9) is a selective agonist for α2-adrenergic receptor (α2A-AR) with EC50 of 0.23 nM. α2A-AR agonist 1 exhibits a hypnotic effect, with ED50 of 0.138 mg/kg in the loss of righting reflex (LORR) experiment. α2A-AR agonist 1 exhibits metabolic stability in mouse liver microsomes[1].

Formula: C12H11BrN2O

References: [1]Lv X, et al., Designing Chromane Derivatives as α2A-Adrenoceptor Selective Agonists via Conformation Constraint. J Med Chem. 2024 Jun 18.

CAS Number: 2971825-58-6

Molecular Weight: 279.13

Research Area: Cancer

Target: Adrenergic Receptor

• SKU: MEXHY-162620-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-162620-0
• Package Unit: Get quote
• Quantity Unit: STK