Product Description: Centanafadine is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively.
Applications: Metabolism-protein/nucleotide metabolism
Formula: C15H15N
References: [1]Bymaster FP, et al. Pharmacological characterization of the norepinephrine and dopamine reuptake inhibitor EB-1020: implications for treatment of attention-deficit hyperactivity disorder. Synapse. 2012 Jun;66(6):522-32.
CAS Number: 924012-43-1
Molecular Weight: 209.29
Compound Purity: 99.62
Research Area: Neurological Disease; Endocrinology
Solubility: DMSO : 125 mg/mL (ultrasonic)
Target: Adrenergic Receptor;Dopamine Transporter;Serotonin Transporter