Product Description: GRA Ex-25 is an inhibitor of glucagon receptor, with IC50 of 56 and 55 nM for rat and human glucagon receptors, respectively.
Applications: Metabolism-sugar/lipid metabolism
Formula: C29H36F3N3O5
References: [1]Kurukulasuriya R, et al. Biaryl amide glucagon receptor antagonists. Bioorg Med Chem Lett. 2004 May 3;14(9):2047-50./[2]Kurukulasuriya R, et al. Biaryl amide glucagon receptor antagonists. Bioorg Med Chem Lett. 2004 May 3;14(9):2047-50.
CAS Number: 307983-31-9
Molecular Weight: 563.6084496
Compound Purity: 98.59
Research Area: Metabolic Disease
Solubility: DMSO : ≥ 32 mg/mL
Target: GCGR