hMC1R agonist 1, CAS 3028881-87-7

Product Description: (EC50=3 nM). hMC1R agonist 1 shows at least 300-fold selectivity for hMC1R over hMC3R (b>EC50=902 nM), hMC4R (b>EC50=915 nM), and hMC5R (b>EC50=>1000 nM). hMC1R agonist 1 has the potential for the therapeutic intervention of melanocortin family[1].

Applications: COVID-19-immunoregulation

Formula: C54H70N14O8S2

References: [1]Nafie MS, et al. Exploration of novel VEGFR2 tyrosine kinase inhibitors via design and synthesis of new alkylated indolyl-triazole Schiff bases for targeting breast cancer. Bioorg Chem. 2022; 122:105708.

CAS Number: 3028881-87-7

Molecular Weight: 1107.35

Compound Purity: 99.37

Research Area: Inflammation/Immunology

Solubility: DMSO : 100 mg/mL (ultrasonic)

Target: Melanocortin Receptor

• SKU: MEXHY-P99004-10
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-P99004-10
• Green Labware: No
• Package Unit: 10 mg
• Quantity Unit: STK