MOR agonist-4

Product Description: MOR agonist-4 (2d) is a G protein signaling-biased Kappa opioid receptor (KOR) agonist with an EC50 value of 11 nM. MOR agonist-4 contains an electron withdrawing CF3 group and a bias factor of 38 based on triazole. MOR agonist-4 is used in the research of pruritis and analgesia[1].

Formula: C22H19F3N4S

References: [1]Trojniak AE, et al. Synthesis and evaluation of 3,4,5-trisubstituted triazoles as G protein-biased kappa opioid receptor agonists[J]. Eur J Med Chem. 2024 Jun 27;276:116627.

Molecular Weight: 428.47

Research Area: Others

Target: Opioid Receptor

• SKU: MEXHY-161812-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-161812-0
• Package Unit: Get quote
• Quantity Unit: STK