N-myristoyl-RKRTLRRL, CAS 152246-40-7

Product Description: N-myristoyl-RKRTLRRL inhibits binding of PKC substrates. N-myristoyl-RKRTLRRL inhibits Ca2+- and phosphatidylserine (PS)-dependent histone phosphorylation with IC50 of 5 μM. histone phosphorylation with IC50 of 80 μM[1][2].

Applications: Cancer-Kinase/protease

Formula: C60H117N21O11

References: [1]David K Crockett, et al. Identification of proteins from formalin-fixed paraffin-embedded cells by LC-MS/MS. Lab Invest. 2005 Nov;85(11):1405-15./[2]C A O'Brian, et al. A novel N-myristylated synthetic octapeptide inhibits protein kinase C activity and partially reverses murine fibrosarcoma cell resistance to Adriamycin. Invest New Drugs. 1991 May;9(2):169-79.

CAS Number: 152246-40-7

Molecular Weight: 1308.71

Compound Purity: 99.37

Research Area: cancer

Solubility: DMSO : 50 mg/mL (ultrasonic)

Target: PKC

• SKU: MEXHY-P5988-5
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-P5988-5
• Green Labware: No
• Package Unit: 5 mg
• Quantity Unit: STK