Resomelagon (methanesulfonate), CAS 2933183-20-9

Product Description: Resomelagon methanesulfonate (AP1189 methanesulfonate) is the methanesulfonate salt form of Resomelagon (HY-147301). Resomelagon methanesulfonate is an orally active melanocortin receptor (MR) agonist. Resomelagon methanesulfonate induces ERK1/2 phosphorylation and Ca2+ mobilization. Resomelagon methanesulfonate exhibits anti-inflammatory activity in mouse peritonitis and peritonitis model. Resomelagon methanesulfonate can be used for obesity and chronic inflammation research[1][2].

Applications: COVID-19-immunoregulation

Formula: C15H18N6O5S

References: [1]Montero-Melendez T, et, al. Biased agonism as a novel strategy to harness the proresolving properties of melanocortin receptors without eliciting melanogenic effects. J Immunol. 2015 Apr 1;194(7):3381-8./[2]WHO Drug Information. International Nonproprietary Names for Pharmaceutical.

CAS Number: 2933183-20-9

Molecular Weight: 394.41

Research Area: Inflammation/Immunology

Target: ERK;Melanocortin Receptor

• SKU: MEXHY-147301B-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-147301B-0
• Package Unit: Get quote
• Quantity Unit: STK