Roluperidone, CAS 359625-79-9

Product Description: Roluperidone (CYR-101) is a novel cyclic amide derivative that has high equipotent affinities for 5-HT2A and sigma-2 receptors (Ki of 7.53 nM and 8.19 nM for 5-HT2A and sigma-2, respectively).

Applications: Neuroscience-Neuromodulation

Formula: C22H23FN2O2

References: [1]Davidson M, et al. Efficacy and Safety of MIN-101: A 12-Week Randomized, Double-Blind, Placebo-Controlled Trial of a New Drug in Development for the Treatment of Negative Symptoms in Schizophrenia. Am J Psychiatry. 2017 Jul 28:appiajp201717010122.

CAS Number: 359625-79-9

Molecular Weight: 366.43

Compound Purity: 99.86

Research Area: Neurological Disease

Solubility: DMSO : 33.33 mg/mL (ultrasonic)

Target: 5-HT Receptor;Sigma Receptor

• SKU: MEXHY-19469-25
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-19469-25
• Package Unit: 25 mg
• Quantity Unit: STK