TAS2940 (fumarate), CAS 2758034-98-7

Product Description: TAS2940 fumarate is a brain-penetrable, orally active, irreversible and selective pan-ERBB inhibitor. TAS2940 fumarate against wild-type HER2, HER2 V777L, and A775_G776insYVMA with IC50 values of 5.6 nM, 2.1 nM, and 1.0 nM, respectively. TAS2940 fumarate can be used for the study of tumors with HER2 and EGFR aberrations[1].

Formula: C32H34N6O6

References: [1]Kei Oguchi, et al. TAS2940, a novel brain-penetrable pan-ERBB inhibitor, for tumors with HER2 and EGFR aberrations. Cancer Sci. 2023 Feb;114(2):654-664.

CAS Number: 2758034-98-7

Molecular Weight: 598.65

Research Area: Cancer

Target: EGFR

• SKU: MEXHY-153856A-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-153856A-0
• Package Unit: Get quote
• Quantity Unit: STK