TGR5 agonist 5

Product Description: TGR5 agonist 5 (compound K91) is a potent agonist of TGR5, with EC50s of 19 μM and 30 μM in CRE-Luciferase assay anf cAMP accumulation assay, respectively[1].

Formula: C22H26N2O2

References: [1]M Giovanna E Papadopoulos, et al. Discovery and characterization of small-molecule TGR5 ligands with agonistic activity. Eur J Med Chem. 2024 Jun 28:276:116616.

Molecular Weight: 350.45

Research Area: Others

Target: G protein-coupled Bile Acid Receptor 1

• SKU: MEXHY-161817-0
• Manufacturer: MedChemExpress
• Manufacturer SKU: HY-161817-0
• Package Unit: Get quote
• Quantity Unit: STK