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Biological Activity: Entacapone potently inhibits rat liver total COMT with IC50 and Ki values of 20.1 nM and 10.7 nM respectively. The IC50 values of entacapone against rat liver soluble COMT (S-COMT) and rat liver membrane-bound COMT (MB-COMT) are 14.3 nM and 73.3 nM respectively.
CAS Number: 130929-57-6
Description: Entacapone is a second-generation catechol-O-methyltransferase (COMT) inhibitor
Purity: ≥98% by HPLC
Solubility: Soluble in DMSO 61 mg/ml, water <1 mg/ml, ethanol 2 mg/ml
Storage Stability: Store at or below -20°C. Solid form is stable at least 12 months from date of receipt, when stored as directed. Do not store aqueous solutions for more than one day.
Target: COMT
Biosafety Level: Not applicable (BSL-1)
References: Forsberg M, et al. J Pharmacol Exp Ther. 2003 Feb;304(2):498-506.
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