FMF-04-159-2, CAS 2364489-81-4

Formulation: A solid

Formal Name: N-[1-[[3-[[(2E)-4-(dimethylamino)-1-oxo-2-buten-1-yl]amino]phenyl]sulfonyl]-4-piperidinyl]-4-[(2,4,6-trichlorobenzoyl)amino]-1H-pyrazole-3-carboxamide

Purity: ≥95%

Formula Markup: C28H30Cl3N7O5S

Formula Weight: 683

Shelf life (days): 1460

CAS Number: 2364489-81-4

Notes: FMF-04-159-2 is an inhibitor of TAIRE family kinases.{67700} It binds to Cdk14 and Cdk16 (IC50s = 88 and 10.1 nM, respectively) and selectively inhibits Cdk14, Cdk16, Cdk17, and Cdk18 over a panel of 16 additional kinases at 1 µM but does inhibit Cdk2 and Cdk10 by greater than 70% at 1 µM.

• SKU: CAY39989-1
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 39989-1
• Package Unit: 1 mg
• Quantity Unit: STK