GSK620, CAS 2088410-46-0

Formulation: A solid

Formal Name: N5-cyclopropyl-1,2-dihydro-N3-methyl-2-oxo-1-(phenylmethyl)-3,5-pyridinedicarboxamide

Purity: ≥98%

Formula Markup: C18H19N3O3

CAS Number: 2088410-46-0

Notes: GSK620 is a bromodomain and extra terminal domain family of proteins (BET) bromodomain 2 (BD2) inhibitor (IC50s = 316.2, 79.4, 79.4, and 199.5 nM for BRD2, BRD3, BRD4, and BRDT BD2, respectively).{68741} It is selective for BD2 in bromodomain-containing protein 2 (BRD2), BRD3, BRD4, and BRDT over BD1 in the same BRDs (IC50s = >15,000 nM for all). GSK620 inhibits LPS-induced chemokine (C-C motif) ligand 1 (CCL1) production in isolated human whole blood (IC50 = 794.3 nM).

• SKU: CAY36139-50
• Manufacturer: Cayman Chemical
• Manufacturer SKU: 36139-50
• Package Unit: 50 mg
• Quantity Unit: STK